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Givinostat
CAS No. 732302-99-7
Givinostat ( ITF2357 )
产品货号. M15799 CAS No. 732302-99-7
Givinostat hydrochloride monohydrate is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively.
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥583 | 有现货 |
|
| 10MG | ￥1037 | 有现货 |
|
| 25MG | ￥2049 | 有现货 |
|
| 50MG | ￥3750 | 有现货 |
|
| 100MG | ￥5532 | 有现货 |
|
| 500MG | ￥11745 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Givinostat
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Givinostat hydrochloride monohydrate is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively.
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产品描述Givinostat hydrochloride monohydrate is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively.
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同义词ITF2357
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HD1-A; HD1-B; HD2
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研究领域Inflammation/Immunology
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适应症——
化学信息
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CAS Number732302-99-7
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分子量475.97
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分子式CHClNO
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纯度>98%(HPLC)
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溶解度DMSO:95 mg/mL (199.59 mM); Ethanol:3 mg/mL (6.3 mM); Water:<1 mg/mL (<1 mM)
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SMILESO=C(OCC1=CC=C2C=C(CN(CC)CC)C=CC2=C1)NC3=CC=C(C(NO)=O)C=C3.[H]Cl.O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Li S, et al. Specific inhibition of histone deacetylase 8 reduces gene expression and production of proinflammatory cytokines in vitro and in vivo. J Biol Chem. 2015 Jan 23;290(4):2368-78.
产品手册
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